International Union of Pharmacology. XV. Subtypes of gamma-aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function.
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- Authors
- Barnard, E A; Skolnick, P; Olsen, R W; Mohler, H; Sieghart, W; Biggio, G; Braestrup, C; Bateson, A N; Langer, S Z
- Year
- 1998
- Journal
- Pharmacological reviews
- PMID
- 9647870
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| Search for Ξ±3Ξ²β/βΞ³2 subtype selective ligands that are stable on human liver microsomes. | Namjoshi OA et al. | β | 2013 | β |
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| The effects of chronic taurine supplementation on motor learning. | Santora A et al. | β | 2013 | β |
| The parvalbumin-positive interneurons in the mouse dentate gyrus express GABAA receptor subunits Ξ±1, Ξ²2, and Ξ΄ along their extrasynaptic cell membrane. | Milenkovic I et al. | β | 2013 | β |
| Yellow fluorescent protein-based assay to measure GABA(A) channel activation and allosteric modulation in CHO-K1 cells. | Johansson T et al. | β | 2013 | β |
| A common variant in ERBB4 regulates GABA concentrations in human cerebrospinal fluid. | Luykx JJ et al. | β | 2012 | β |
| Acute behavioural responses to nicotine and nicotine withdrawal syndrome are modified in GABA(B1) knockout mice. | Varani AP et al. | β | 2012 | β |
| Adolescent female rats exhibiting activity-based anorexia express elevated levels of GABA(A) receptor Ξ±4 and Ξ΄ subunits at the plasma membrane of hippocampal CA1 spines. | Aoki C et al. | β | 2012 | β |
| Anxioselective anxiolytics: on a quest for the Holy Grail. | Skolnick P | β | 2012 | β |
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| GABRG1 and GABRA2 variation associated with alcohol dependence in African Americans. | Ittiwut C et al. | β | 2012 | β |
| General anesthesia mediated by effects on ion channels. | Zhou C et al. | β | 2012 | β |
| Genetics of GABAergic signaling in nicotine and alcohol dependence. | Cui WY et al. | β | 2012 | β |
| Gephyrin, the enigmatic organizer at GABAergic synapses. | Tretter V et al. | β | 2012 | β |
| Histaminergic pharmacology of homo-oligomeric Ξ²3 Ξ³-aminobutyric acid type A receptors characterized by surface plasmon resonance biosensor technology. | Seeger C et al. | β | 2012 | β |
| Homocysteine alters cerebral microvascular integrity and causes remodeling by antagonizing GABA-A receptor. | Lominadze D et al. | β | 2012 | β |
| Hydroxylated biphenyl derivatives are positive modulators of human GABA(A) receptors. | Paola Mascia M et al. | β | 2012 | β |
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| Knockout of the Ξ³-aminobutyric acid receptor subunit Ξ±4 reduces functional Ξ΄-containing extrasynaptic receptors in hippocampal pyramidal cells at the onset of puberty. | Sabaliauskas N et al. | β | 2012 | β |
| Low nanomolar GABA effects at extrasynaptic Ξ±4Ξ²1/Ξ²3Ξ΄ GABA(A) receptor subtypes indicate a different binding mode for GABA at these receptors. | Karim N et al. | β | 2012 | β |
| Structure, function, and modulation of GABA(A) receptors. | Sigel E et al. | β | 2012 | β |
| Tlx1/3 and Ptf1a control the expression of distinct sets of transmitter and peptide receptor genes in the developing dorsal spinal cord. | Guo Z et al. | β | 2012 | β |
| Widespread abnormality of the Ξ³-aminobutyric acid-ergic system in Tourette syndrome. | Lerner A et al. | β | 2012 | β |
| Absorption, excretion, and metabolism of a potential GABA-A Ξ±2/3 receptor modulator in rats. | Guo J et al. | β | 2011 | β |
| Anxiolytic activity of pyridoindole derivatives SMe1EC2 and SMe1M2: behavioral analysis using rat model. | SedlΓ‘ΔkovΓ‘ N et al. | β | 2011 | β |
| Central and Peripheral GABA(A) Receptor Regulation of the Heart Rate Depends on the Conscious State of the Animal. | Bentzen BH et al. | β | 2011 | β |
| GABAA receptor open-state conformation determines non-competitive antagonist binding. | Chen L et al. | β | 2011 | β |
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| Hooked on benzodiazepines: GABAA receptor subtypes and addiction. | Tan KR et al. | β | 2011 | β |
| HZ166, a novel GABAA receptor subtype-selective benzodiazepine site ligand, is antihyperalgesic in mouse models of inflammatory and neuropathic pain. | Di Lio A et al. | β | 2011 | β |
| Implications for treatment: GABAA receptors in aging, Down syndrome and Alzheimer's disease. | Rissman RA et al. | β | 2011 | β |
| Inhibition of learning and memory by general anesthetics. | Wang DS et al. | β | 2011 | β |
| Light it up: highly efficient multigene delivery in mammalian cells. | Trowitzsch S et al. | β | 2011 | β |
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| Neurosteroid modulation of benzodiazepine-sensitive GABAA tonic inhibition in supraoptic magnocellular neurons. | Jo JY et al. | β | 2011 | β |
| Neurosteroidogenesis is required for the physiological response to stress: role of neurosteroid-sensitive GABAA receptors. | Sarkar J et al. | β | 2011 | β |
| Neurovascular interaction and the pathophysiology of diabetic retinopathy. | Qian H et al. | β | 2011 | β |
| New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds. | Anzini M et al. | β | 2011 | β |
| Potentiation and inhibition of glycine receptors by tutin. | Fuentealba J et al. | β | 2011 | β |
| Prediction of GABAA receptor proteins using the concept of Chou's pseudo-amino acid composition and support vector machine. | Mohabatkar H et al. | β | 2011 | β |
| Seizure susceptibility in polymicrogyria: clinical and experimental approaches. | Takano T | β | 2011 | β |
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| The sedative but not the memory-blocking properties of ethanol are modulated by Ξ±5-subunit-containing Ξ³-aminobutyric acid type A receptors. | Martin LJ et al. | β | 2011 | β |
| Thymoquinone produced antianxiety-like effects in mice through modulation of GABA and NO levels. | Gilhotra N et al. | β | 2011 | β |
| Tolerance to allopregnanolone with focus on the GABA-A receptor. | Turkmen S et al. | β | 2011 | β |
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| Benzodiazepine modulation of the rat GABAA receptor Ξ±4Ξ²3Ξ³2L subtype expressed in Xenopus oocytes. | You H et al. | β | 2010 | β |
| Bioactivity-guided isolation of GABA(A) receptor modulating constituents from the rhizomes of Actaea racemosa. | Cicek SS et al. | β | 2010 | β |
| Design, synthesis, and subtype selectivity of 3,6-disubstituted Ξ²-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse. | Yin W et al. | β | 2010 | β |
| Distinct Ξ± subunit variations of the hypothalamic GABAA receptor triplets (Ξ±Ξ²Ξ³) are linked to hibernating state in hamsters. | AlΓ² R et al. | β | 2010 | β |
| Diversity of structure and function of alpha1alpha6beta3delta GABAA receptors: comparison with alpha1beta3delta and alpha6beta3delta receptors. | Baur R et al. | β | 2010 | β |
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| GABRA2 and alcohol use disorders: no evidence of an association in an Italian case-control study. | Onori N et al. | β | 2010 | β |
| GABRR1 and GABRR2, encoding the GABA-A receptor subunits rho1 and rho2, are associated with alcohol dependence. | Xuei X et al. | β | 2010 | β |
| Improved reversal learning and working memory and enhanced reactivity to novelty in mice with enhanced GABAergic innervation in the dentate gyrus. | Morellini F et al. | β | 2010 | β |
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| Molecular mechanisms of general anesthesia. | Son Y | β | 2010 | β |
| New insights into the molecular mechanisms of general anaesthetics. | Chau PL | β | 2010 | β |
| Prototypic GABA(A) receptor agonist muscimol acts preferentially through forebrain high-affinity binding sites. | Chandra D et al. | β | 2010 | β |
| Role of central neurotransmission and chemoreception on airway control. | Kc P et al. | β | 2010 | β |
| The effects of zolpidem treatment and withdrawal on the in vitro expression of recombinant alpha1beta2gamma2s GABA(A) receptors expressed in HEK 293 cells. | VlainiΔ J et al. | β | 2010 | β |
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| Zolpidem modulation of phasic and tonic GABA currents in the rat dorsal motor nucleus of the vagus. | Gao H et al. | β | 2010 | β |
| Age- and gender-related differences in GABAA receptor-mediated postsynaptic currents in GABAergic neurons of the substantia nigra reticulata in the rat. | Chudomel O et al. | β | 2009 | β |
| Allosteric modulation by benzodiazepines of GABA-gated chloride channels of an identified insect motor neurone. | Buckingham SD et al. | β | 2009 | β |
| Altering the relative abundance of GABA A receptor subunits changes GABA- and ethanol-responses in Xenopus oocytes. | Hurley JH et al. | β | 2009 | β |
| A nomenclature for ligand-gated ion channels. | Collingridge GL et al. | β | 2009 | β |
| Changes in expression and function of extrasynaptic GABAA receptors in the rat hippocampus during pregnancy and after delivery. | Sanna E et al. | β | 2009 | β |
| Complete sequencing of GABAA receptor subunit beta 3 by a rapid technique following in-gel digestion of the protein. | Kang SU et al. | β | 2009 | β |
| Current status of inverse agonism at serotonin2A (5-HT2A) and 5-HT2C receptors. | Aloyo VJ et al. | β | 2009 | β |
| Distinct structural changes in the GABAA receptor elicited by pentobarbital and GABA. | Muroi Y et al. | β | 2009 | β |
| Docking of 1,4-benzodiazepines in the alpha1/gamma2 GABA(A) receptor modulator site. | Berezhnoy D et al. | β | 2009 | β |
| Effects of isopulegol on pentylenetetrazol-induced convulsions in mice: possible involvement of GABAergic system and antioxidant activity. | Silva MI et al. | β | 2009 | β |
| Expression quantitative trait loci and genetic regulatory network analysis reveals that Gabra2 is involved in stress responses in the mouse. | Dai J et al. | β | 2009 | β |
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| GABAA receptor alpha5 subunits contribute to GABAA,slow synaptic inhibition in mouse hippocampus. | Zarnowska ED et al. | β | 2009 | β |
| GABA(A) receptors and their associated proteins: implications in the etiology and treatment of schizophrenia and related disorders. | Charych EI et al. | β | 2009 | β |
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| GABRG1 and GABRA2 as independent predictors for alcoholism in two populations. | Enoch MA et al. | β | 2009 | β |
| Gel-based mass spectrometric analysis of a strongly hydrophobic GABAA-receptor subunit containing four transmembrane domains. | Kang SU et al. | β | 2009 | β |
| Homology modeling of human alpha 1 beta 2 gamma 2 and house fly beta 3 GABA receptor channels and Surflex-docking of fipronil. | Cheng J et al. | β | 2009 | β |
| Indiplon in the management of insomnia. | Lemon MD et al. | β | 2009 | β |
| Investigation of ethanol-induced impairment of spatial memory in gamma2 heterozygous knockout mice. | Berry RB et al. | β | 2009 | β |
| Plasticity and function of extrasynaptic GABA(A) receptors during pregnancy and after delivery. | Mostallino MC et al. | β | 2009 | β |
| Quantitative analyses of [ΒΉΒΉC]Ro15-4513 binding to subunits of GABAA/benzodiazepine receptor in the living human brain. | Asai Y et al. | β | 2009 | β |
| Similar anxiolytic-like effects following intra-amygdala infusions of benzodiazepine receptor agonist and antagonist: evidence for the release of an endogenous benzodiazepine inverse agonist in mice exposed to elevated plus-maze test. | Barbalho CA et al. | β | 2009 | β |
| The alpha5(H105R) mutation impairs alpha5 selective binding properties by altered positioning of the alpha5 subunit in GABAA receptors containing two distinct types of alpha subunits. | Balic E et al. | β | 2009 | β |
| The interaction of sildenafil with the anticonvulsant effect of diazepam. | Gholipour T et al. | β | 2009 | β |
| The regulation of neuronal gene expression by alcohol. | Pignataro L et al. | β | 2009 | β |
| Unanticipated structural and functional properties of delta-subunit-containing GABAA receptors. | Kaur KH et al. | β | 2009 | β |
| Unraveling the molecular mechanisms of alcohol dependence. | Kalsi G et al. | β | 2009 | β |
| 6,3'-Dinitroflavone is a low efficacy modulator of GABA(A) receptors. | Furtmueller R et al. | β | 2008 | β |
| alpha1beta2delta, a silent GABAA receptor: recruitment by tracazolate and neurosteroids. | Zheleznova N et al. | β | 2008 | β |
| Antimalarial drugs inhibit human 5-HT(3) and GABA(A) but not GABA(C) receptors. | Thompson AJ et al. | β | 2008 | β |
| Assessment of GABAA benzodiazepine receptor (GBzR) sensitivity in patients with alcohol dependence. | Taylor C et al. | β | 2008 | β |
| Attenuation of morphine withdrawal signs by muscimol in the locus coeruleus of rats. | Mirzaii-Dizgah I et al. | β | 2008 | β |
| Behavioral effects of 6-bromoflavanone and 5-methoxy-6,8-dibromoflavanone as anxiolytic compounds. | Ognibene E et al. | β | 2008 | β |
| Current and prospective pharmacological targets in relation to antimigraine action. | Mehrotra S et al. | β | 2008 | β |
| Developmental maturation of synaptic and extrasynaptic GABAA receptors in mouse thalamic ventrobasal neurones. | Peden DR et al. | β | 2008 | β |
| Differential effects of diazepam treatment and withdrawal on recombinant GABAA receptor expression and functional coupling. | Svob Strac D et al. | β | 2008 | β |
| Estimating the efficiency of benzodiazepines on GABA(A) receptors comprising gamma1 or gamma2 subunits. | Baburin I et al. | β | 2008 | β |
| GABA-A2 receptor subunit gene (GABRA2) polymorphisms and risk for alcohol dependence. | Soyka M et al. | β | 2008 | β |
| GABA(A) receptor properties in catastrophic infantile epilepsy. | Jansen LA et al. | β | 2008 | β |
| GABA(A) receptors and alcohol. | Lobo IA et al. | β | 2008 | β |
| GABA(A) receptors in normal development and seizures: friends or foes? | Galanopoulou AS | β | 2008 | β |
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| GABA(A) receptor trafficking and its role in the dynamic modulation of neuronal inhibition. | Jacob TC et al. | β | 2008 | β |
| Guest editor's note. | Reynolds DS et al. | β | 2008 | β |
| HPLC-based activity profiling approach for the discovery of GABAA receptor ligands using an automated two microelectrode voltage clamp assay on Xenopus oocytes. | Kim HJ et al. | β | 2008 | β |
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| International Union of Pharmacology. LXX. Subtypes of gamma-aminobutyric acid(A) receptors: classification on the basis of subunit composition, pharmacology, and function. Update. | Olsen RW et al. | β | 2008 | β |
| Interpopulation linkage disequilibrium patterns of GABRA2 and GABRG1 genes at the GABA cluster locus on human chromosome 4. | Ittiwut C et al. | β | 2008 | β |
| Investigating the putative binding-mode of GABA and diazepam within GABA A receptor using molecular modeling. | Ci S et al. | β | 2008 | β |
| Investigation of gamma-aminobutyric acid (GABA) A receptors genes and migraine susceptibility. | Fernandez F et al. | β | 2008 | β |
| Juvenile stress-induced alteration of maturation of the GABAA receptor alpha subunit in the rat. | Jacobson-Pick S et al. | β | 2008 | β |
| Menthol shares general anesthetic activity and sites of action on the GABA(A) receptor with the intravenous agent, propofol. | Watt EE et al. | β | 2008 | β |
| Molecular dynamics simulations of GABA binding to the GABAC receptor: the role of Arg104. | Melis C et al. | β | 2008 | β |
| Molecular mechanisms supporting a paracrine role of GABA in rat adrenal medullary cells. | Matsuoka H et al. | β | 2008 | β |
| Neuroactive steroids and GABAA receptor plasticity in the brain of the WAG/Rij rat, a model of absence epilepsy. | Pisu MG et al. | β | 2008 | β |
| Normal acute behavioral responses to moderate/high dose ethanol in GABAA receptor alpha 4 subunit knockout mice. | Chandra D et al. | β | 2008 | β |
| Pharmacological Properties of DOV 315,090, an ocinaplon metabolite. | Berezhnoy D et al. | β | 2008 | β |
| Regional differences in the decay kinetics of GABA(A) receptor-mediated miniature IPSCs in the dorsal horn of the rat spinal cord are determined by mitochondrial transport of cholesterol. | Inquimbert P et al. | β | 2008 | β |
| Relationship between neuronal vulnerability and potassium-chloride cotransporter 2 immunoreactivity in hippocampus following transient forebrain ischemia. | Papp E et al. | β | 2008 | β |
| Structural determinants for antagonist pharmacology that distinguish the rho1 GABAC receptor from GABAA receptors. | Zhang J et al. | β | 2008 | β |
| Surface expression of GABAA receptors is transcriptionally controlled by the interplay of cAMP-response element-binding protein and its binding partner inducible cAMP early repressor. | Hu Y et al. | β | 2008 | β |
| Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site. | Jansen M et al. | β | 2008 | β |
| The role of GABA(A) receptors in the development of alcoholism. | Enoch MA | β | 2008 | β |
| The role of GABAergic transmission in the dentate gyrus on acquisition, consolidation and retrieval of an inhibitory avoidance learning and memory task in the rat. | Shahidi S et al. | β | 2008 | β |
| The role of transcriptional and translational mechanisms in flumazenil-induced up-regulation of recombinant GABA(A) receptors. | JazvinsΔak Jembrek M et al. | β | 2008 | β |
| Tonically active inhibition selectively controls feedforward circuits in mouse barrel cortex. | Krook-Magnuson EI et al. | β | 2008 | β |
| Translational aspects of pharmacological research into anxiety disorders: the stress-induced hyperthermia (SIH) paradigm. | Vinkers CH et al. | β | 2008 | β |
| [3H] muscimol receptors sites in the carp (Cyprinus carpio L.) brain: binding assay and autoradiographic distribution. | Pirone A et al. | β | 2007 | β |
| 6,2'-Dihydroxyflavone, a subtype-selective partial inverse agonist of GABAA receptor benzodiazepine site. | Wang F et al. | β | 2007 | β |
| A conserved tyrosine in the beta2 subunit M4 segment is a determinant of gamma-aminobutyric acid type A receptor sensitivity to propofol. | Richardson JE et al. | β | 2007 | β |
| Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors. | PericiΔ D et al. | β | 2007 | β |
| Anticonvulsant actions of deoxycorticosterone. | Perez-Cruz C et al. | β | 2007 | β |
| A single point mutation of the GABA(A) receptor alpha5-subunit confers fluoxetine sensitivity. | Derry JM et al. | β | 2007 | β |
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| Benzodiazepine receptor agonists affect both binding and gating of recombinant alpha1beta2gamma2 gamma-aminobutyric acid-A receptors. | Mercik K et al. | β | 2007 | β |
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| Changes in the function of the inhibitory neurotransmitter system in the rat brain following subchronic inhalation exposure to 1-bromopropane. | Ueno S et al. | β | 2007 | β |
| Characterization of [35S]t-butylbicyclophosphorothionate ([35S]TBPS) binding to GABAA receptors in postmortem human brain. | Atack JR et al. | β | 2007 | β |
| Chronic progesterone treatment augments while dehydroepiandrosterone sulphate prevents tolerance to ethanol anxiolysis and withdrawal anxiety in rats. | Sharma AN et al. | β | 2007 | β |
| CNS 7056: a novel ultra-short-acting Benzodiazepine. | Kilpatrick GJ et al. | β | 2007 | β |
| Colocalization of synaptic GABA(C)-receptors with GABA (A)-receptors and glycine-receptors in the rodent central nervous system. | Frazao R et al. | β | 2007 | β |
| Comparative effects of nonselective and subtype-selective gamma-aminobutyric acidA receptor positive modulators in the rat-conditioned emotional response test. | Mathiasen LS et al. | β | 2007 | β |
| Contribution of specific binding to the central benzodiazepine site to the brain concentrations of two novel benzodiazepine site ligands. | Pike A et al. | β | 2007 | β |
| Differential expression of gamma-aminobutyric acid receptor A (GABA(A)) and effects of homocysteine. | Tyagi N et al. | β | 2007 | β |
| Does ethanol act preferentially via selected brain GABAA receptor subtypes? the current evidence is ambiguous. | Korpi ER et al. | β | 2007 | β |
| Etomidate and propofol-hyposensitive GABAA receptor beta3(N265M) mice show little changes in acute alcohol sensitivity but enhanced tolerance and withdrawal. | Sanchis-Segura C et al. | β | 2007 | β |
| Exploring ligand recognition and ion flow in comparative models of the human GABA type A receptor. | Mokrab Y et al. | β | 2007 | β |
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| GABAA and glycine receptor-mediated transmission in rat lamina II neurones: relevance to the analgesic actions of neuroactive steroids. | Mitchell EA et al. | β | 2007 | β |
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| Involvement of chloride channel coupled GABA(C) receptors in the peripheral antinociceptive effect induced by GABA(C) receptor agonist cis-4-aminocrotonic acid. | Reis GM et al. | β | 2007 | β |
| Mapping the contribution of beta3-containing GABAA receptors to volatile and intravenous general anesthetic actions. | Zeller A et al. | β | 2007 | β |
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| New insight into the role of the beta3 subunit of the GABAA-R in development, behavior, body weight regulation, and anesthesia revealed by conditional gene knockout. | Ferguson C et al. | β | 2007 | β |
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| Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities. | Hadley SH et al. | β | 2007 | β |
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| The amygdala regulates the antianxiety sensitization effect of flumazenil during repeated chronic ethanol or repeated stress. | Knapp DJ et al. | β | 2007 | β |
| The GABAA receptor: a novel target for treatment of fragile X? | D'Hulst C et al. | β | 2007 | β |
| The role of the GABRA2 polymorphism in multiplex alcohol dependence families with minimal comorbidity: within-family association and linkage analyses. | Matthews AG et al. | β | 2007 | β |
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| Age-related alterations in GABA(A) receptor subunits in the nonhuman primate hippocampus. | Rissman RA et al. | β | 2006 | β |
| Alcohol-sensitive GABA receptors and alcohol antagonists. | Paul SM | β | 2006 | β |
| An interaction between benzodiazepines and neuroactive steroids at GABA A receptors in cultured hippocampal neurons. | Ahboucha S et al. | β | 2006 | β |
| An inversion inv(4)(p12-p15.3) in autistic siblings implicates the 4p GABA receptor gene cluster. | Vincent JB et al. | β | 2006 | β |
| Autoradiographic localization and binding study of benzodiazepines receptor sites in carp brain (Cyprinus carpio L.). | Pirone A et al. | β | 2006 | β |
| Changes in expression of GABAA alpha4 subunit mRNA in the brain under anesthesia induced by volatile and intravenous anesthetics. | Sekine S et al. | β | 2006 | β |
| Changes in neocortical and hippocampal GABAA receptor subunit distribution during brain maturation and aging. | Yu ZY et al. | β | 2006 | β |
| Comparative cue generalization profiles of L-838, 417, SL651498, zolpidem, CL218,872, ocinaplon, bretazenil, zopiclone, and various benzodiazepines in chlordiazepoxide and zolpidem drug discrimination. | Mirza NR et al. | β | 2006 | β |
| Compensatory alteration of inhibitory synaptic circuits in cerebellum and thalamus of gamma-aminobutyric acid type A receptor alpha1 subunit knockout mice. | Kralic JE et al. | β | 2006 | β |
| Contributions of the GABAA receptor alpha6 subunit to phasic and tonic inhibition revealed by a naturally occurring polymorphism in the alpha6 gene. | Santhakumar V et al. | β | 2006 | β |
| Effect of extracellular pH on recombinant alpha1beta2gamma2 and alpha1beta2 GABAA receptors. | Mercik K et al. | β | 2006 | β |
| Evidence that GABA rho subunits contribute to functional ionotropic GABA receptors in mouse cerebellar Purkinje cells. | Harvey VL et al. | β | 2006 | β |
| Expression profiling suggests underexpression of the GABA(A) receptor subunit delta in the fragile X knockout mouse model. | Gantois I et al. | β | 2006 | β |
| GABAA receptor alpha 4 subunits mediate extrasynaptic inhibition in thalamus and dentate gyrus and the action of gaboxadol. | Chandra D et al. | β | 2006 | β |
| GABA receptors ameliorate Hcy-mediated integrin shedding and constrictive collagen remodeling in microvascular endothelial cells. | Shastry S et al. | β | 2006 | β |
| Glutamate and GABA receptors and transporters in the basal ganglia: what does their subsynaptic localization reveal about their function? | Galvan A et al. | β | 2006 | β |
| Graded response to GABA by native extrasynaptic GABA receptors. | Lindquist CE et al. | β | 2006 | β |
| High pH accelerates GABA deactivation on perch-rho1B receptors. | Qian H et al. | β | 2006 | β |
| Identification of amino acid residues important for assembly of GABA receptor alpha1 and gamma2 subunits. | Sarto-Jackson I et al. | β | 2006 | β |
| Imidazenil and diazepam increase locomotor activity in mice exposed to protracted social isolation. | Pinna G et al. | β | 2006 | β |
| Immunofluorescence in brain sections: simultaneous detection of presynaptic and postsynaptic proteins in identified neurons. | Schneider Gasser EM et al. | β | 2006 | β |
| Impact of epsilon and theta subunits on pharmacological properties of alpha3beta1 GABAA receptors expressed in Xenopus oocytes. | Ranna M et al. | β | 2006 | β |
| Methamphetamine induces long-term changes in GABAA receptor alpha2 subunit and GAD67 expression. | Zhang X et al. | β | 2006 | β |
| Molecular and synaptic organization of GABAA receptors in the cerebellum: Effects of targeted subunit gene deletions. | Fritschy JM et al. | β | 2006 | β |
| Neurosteroid modulation of recombinant rat alpha5beta2gamma2L and alpha1beta2gamma2L GABA(A) receptors in Xenopus oocyte. | Rahman M et al. | β | 2006 | β |
| Neurosteroids, GABAA receptors, and ethanol dependence. | Follesa P et al. | β | 2006 | β |
| Normal [3H]flunitrazepam binding to GABAA receptors in the locus coeruleus in major depression and suicide. | Zhu H et al. | β | 2006 | β |
| Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABA(A) alpha5 inverse agonist for cognitive dysfunction. | Jones P et al. | β | 2006 | β |
| Plastic neuronal changes in GABA(A) receptor gene expression induced by progesterone metabolites: in vitro molecular and functional studies. | Biggio F et al. | β | 2006 | β |
| Prenatal alcohol exposure alters GABA(A)alpha5 expression: a mechanism of alcohol-induced learning dysfunction. | Toso L et al. | β | 2006 | β |
| Random assembly of GABA rho1 and rho2 subunits in the formation of heteromeric GABA(C) receptors. | Pan Y et al. | β | 2006 | β |
| Social isolation-induced increase in alpha and delta subunit gene expression is associated with a greater efficacy of ethanol on steroidogenesis and GABA receptor function. | Serra M et al. | β | 2006 | β |
| Structural model for gamma-aminobutyric acid receptor noncompetitive antagonist binding: widely diverse structures fit the same site. | Chen L et al. | β | 2006 | β |
| Synthesis, pharmacology and molecular modeling of N-substituted 2-phenyl-indoles and benzimidazoles as potent GABA(A) agonists. | FalcΓ³ JL et al. | β | 2006 | β |
| The genetics of alcoholism: identifying specific genes through family studies. | Edenberg HJ et al. | β | 2006 | β |
| The lack of bicuculline and picrotoxin influence on midazolam depressant action on brain oxygen consumption. | ObradoviΔ DI et al. | β | 2006 | β |
| A linkage study between the GABAA beta2 and GABAA gamma2 subunit genes and major psychoses. | AmbrΓ³sio AM et al. | β | 2005 | β |
| Alternative splicing and promoter use in the human GABRA2 gene. | Tian H et al. | β | 2005 | β |
| A precritical period for plasticity in visual cortex. | Feller MB et al. | β | 2005 | β |
| Bidirectional effects of benzodiazepine binding site ligands on active avoidance acquisition and retention: differential antagonism by flumazenil and beta-CCt. | SaviΔ MM et al. | β | 2005 | β |
| Charge selectivity of the Cys-loop family of ligand-gated ion channels. | Jensen ML et al. | β | 2005 | β |
| Consequence of the presence of two different beta subunit isoforms in a GABA(A) receptor. | Boulineau N et al. | β | 2005 | β |
| Design, synthesis and biological activity of acyl substituted 3-amino-5-methyl-1,4,5,7-tetrahydropyrazolo[3,4-b]pyridin-6-ones as potential hypnotic drugs. | FalcΓ³ JL et al. | β | 2005 | β |
| Determinants of amentoflavone interaction at the GABA(A) receptor. | Hansen RS et al. | β | 2005 | β |
| Developmental change of GABAergic postsynaptic current in rat periaqueductal gray. | Hahm ET et al. | β | 2005 | β |
| Development of subtype selective GABAA modulators. | Dawson GR et al. | β | 2005 | β |
| Differential expression of gamma-aminobutyric acid--a receptor subunits in rat dorsal and ventral hippocampus. | Sotiriou E et al. | β | 2005 | β |
| Differential GABAA receptor clustering determines GABA synapse plasticity in rat oxytocin neurons around parturition and the onset of lactation. | Koksma JJ et al. | β | 2005 | β |
| Distinct patterns of expression and regulation of GABA receptors containing the delta subunit in cerebellar granule and hippocampal neurons. | Follesa P et al. | β | 2005 | β |
| Don't worry 'B' happy!: a role for GABA(B) receptors in anxiety and depression. | Cryan JF et al. | β | 2005 | β |
| Effects of benzodiazepines receptor agonists on the hypothalamic-pituitary-adrenocortical axis. | Mikkelsen JD et al. | β | 2005 | β |
| Enhancement of benzodiazepine binding sites following chronic treatment with flumazenil. | PericiΔ D et al. | β | 2005 | β |
| Ethyl 2-(4-bromophenyl)-1-(2,4-dichlorophenyl)-1H-4-imidazolecarboxylate is a novel positive modulator of GABAA receptors. | Mascia MP et al. | β | 2005 | β |
| GABA receptors and nitric oxide ameliorate constrictive collagen remodeling in hyperhomocysteinemia. | Shastry S et al. | β | 2005 | β |
| Genetic essential tremor in gamma-aminobutyric acidA receptor alpha1 subunit knockout mice. | Kralic JE et al. | β | 2005 | β |
| Heterogeneity of gamma-aminobutyric acid type A receptors in mitral and tufted cells of the rat main olfactory bulb. | Panzanelli P et al. | β | 2005 | β |
| Influence of the point mutation alpha-1-H101R on the assembly of gamma-aminobutyric acid type A receptors. | Baur R et al. | β | 2005 | β |
| Insomnia in general practice : a consensus report produced by sleep specialists and primary-care physicians in Italy. | Terzano MG et al. | β | 2005 | β |
| Internalized GABA-receptor subunits are transferred to an intracellular pool associated with the postsynaptic density. | van Rijnsoever C et al. | β | 2005 | β |
| Low tolerance and dependence liabilities of etizolam: molecular, functional, and pharmacological correlates. | Sanna E et al. | β | 2005 | β |
| Making sense of GABA(A) receptor subtypes: is a new nomenclature needed? | Nutt DJ | β | 2005 | β |
| Modulation of ethanol withdrawal-induced anxiety-like behavior during later withdrawals by treatment of early withdrawals with benzodiazepine/gamma-aminobutyric acid ligands. | Knapp DJ et al. | β | 2005 | β |
| Neurosteroids: endogenous regulators of the GABA(A) receptor. | Belelli D et al. | β | 2005 | β |
| Novel plant substances acting as beta subunit isoform-selective positive allosteric modulators of GABAA receptors. | Baur R et al. | β | 2005 | β |
| Palatability-dependent appetite and benzodiazepines: new directions from the pharmacology of GABA(A) receptor subtypes. | Cooper SJ | β | 2005 | β |
| Picrotoxin accelerates relaxation of GABAC receptors. | Qian H et al. | β | 2005 | β |
| Selective anxiolysis produced by ocinaplon, a GABA(A) receptor modulator. | Lippa A et al. | β | 2005 | β |
| Selective GABAA alpha5 benzodiazepine inverse agonist antagonizes the neurobehavioral actions of alcohol. | Cook JB et al. | β | 2005 | β |
| Subunit-dependent block by isoflurane of wild-type and mutant alpha(1)S270H GABA(A) receptor currents in Xenopus oocytes. | Hall AC et al. | β | 2005 | β |
| Tandem subunits effectively constrain GABAA receptor stoichiometry and recapitulate receptor kinetics but are insensitive to GABAA receptor-associated protein. | Boileau AJ et al. | β | 2005 | β |
| The GABA rho1 subunit interacts with a cellular retinoic acid binding protein in mammalian retina. | Song XQ et al. | β | 2005 | β |
| Trace fear conditioning is enhanced in mice lacking the delta subunit of the GABAA receptor. | Wiltgen BJ et al. | β | 2005 | β |
| Variations on an inhibitory theme: phasic and tonic activation of GABA(A) receptors. | Farrant M et al. | β | 2005 | β |
| Acute human self-poisoning with the N-phenylpyrazole insecticide fipronil--a GABAA-gated chloride channel blocker. | Mohamed F et al. | β | 2004 | β |
| Affinity of various benzodiazepine site ligands in mice with a point mutation in the GABA(A) receptor gamma2 subunit. | Ogris W et al. | β | 2004 | β |
| A GABAA receptor mutation linked to human epilepsy (gamma2R43Q) impairs cell surface expression of alphabetagamma receptors. | Sancar F et al. | β | 2004 | β |
| A high affinity ligand for GABAA-receptor containing alpha5 subunit antagonizes ethanol's neurobehavioral effects in Long-Evans rats. | McKay PF et al. | β | 2004 | β |
| Alpha 5 subunit-containing GABAA receptors affect the dynamic range of mouse hippocampal kainate-induced gamma frequency oscillations in vitro. | Towers SK et al. | β | 2004 | β |
| Analysis of GABAA receptor function and dissection of the pharmacology of benzodiazepines and general anesthetics through mouse genetics. | Rudolph U et al. | β | 2004 | β |
| Analysis of the set of GABA(A) receptor genes in the human genome. | Simon J et al. | β | 2004 | β |
| Anxioselective anxiolytics: can less be more? | Basile AS et al. | β | 2004 | β |
| Association of SNPs and haplotypes in GABAA receptor beta2 gene with schizophrenia. | Lo WS et al. | β | 2004 | β |
| Behavioral effects of flumazenil in the social conflict test in mice. | UhlΓrovΓ‘ L et al. | β | 2004 | β |
| Bidirectional effects of benzodiazepine binding site ligands in the elevated plus-maze: differential antagonism by flumazenil and beta-CCt. | SaviΔ MM et al. | β | 2004 | β |
| Brain inhibitory mechanisms involved in basic and higher integrated sleep processes. | Gottesmann C | β | 2004 | β |
| Brain regional heterogeneity of pH effects on GABA(A) receptor-associated [35s]TBPS binding. | Uusi-Oukari M et al. | β | 2004 | β |
| Cadmium inhibits GABA-activated ion currents by increasing intracellular calcium level in snail neurons. | MolnΓ‘r G et al. | β | 2004 | β |
| Calcium-independent inhibition of GABA(A) current by caffeine in hippocampal slices. | Taketo M et al. | β | 2004 | β |
| Cellular localization of GABA receptor alpha subunit immunoreactivity in the rat hypothalamus: relationship with neurones containing orexigenic or anorexigenic peptides. | BΓ€ckberg M et al. | β | 2004 | β |
| Characterization of the interaction of indiplon, a novel pyrazolopyrimidine sedative-hypnotic, with the GABAA receptor. | Sullivan SK et al. | β | 2004 | β |
| Chronic exposure of cells expressing recombinant GABAA receptors to benzodiazepine antagonist flumazenil enhances the maximum number of benzodiazepine binding sites. | PericiΔ D et al. | β | 2004 | β |
| Chronic NGF treatment of rat nociceptive DRG neurons in culture facilitates desensitization and deactivation of GABAA receptor-mediated currents. | Fabbro A et al. | β | 2004 | β |
| Chronic prenatal ethanol exposure alters hippocampal GABA(A) receptors and impairs spatial learning in the guinea pig. | Iqbal U et al. | β | 2004 | β |
| Differential effects of ethanol on gamma-aminobutyric acid-A receptor-mediated synaptic currents in congenic strains of inbred long and short-sleep mice. | Proctor WR et al. | β | 2004 | β |
| Differential effects of midazolam on inhibitory postsynaptic currents in CA1 pyramidal cells and dentate gyrus granule cells of rat hippocampal slices. | Kobayashi S et al. | β | 2004 | β |
| Effects of GABA modulators on the repeated acquisition of response sequences in squirrel monkeys. | Campbell UC et al. | β | 2004 | β |
| Effects of status epilepticus on hippocampal GABAA receptors are age-dependent. | Zhang G et al. | β | 2004 | β |
| Ethanol withdrawal-induced up-regulation of the alpha2 subunit of the GABAA receptor and its prevention by diazepam or gamma-hydroxybutyric acid. | Follesa P et al. | β | 2004 | β |
| Four amino acids in the alpha subunits determine the gamma-aminobutyric acid sensitivities of GABAA receptor subtypes. | BΓΆhme I et al. | β | 2004 | β |
| Functional mapping of GABA A receptor subtypes in the amygdala. | Marowsky A et al. | β | 2004 | β |
| GABAA receptors: building the bridge between subunit mRNAs, their promoters, and cognate transcription factors. | Steiger JL et al. | β | 2004 | β |
| GABAA receptor subunit mRNA expression in cultured embryonic and adult human dorsal root ganglion neurons. | Maddox FN et al. | β | 2004 | β |
| GABAA receptor subunits identified in Paramecium by immunofluorescence confocal microscopy. | Ramoino P et al. | β | 2004 | β |
| Genes associated with addiction: alcoholism, opiate, and cocaine addiction. | Kreek MJ et al. | β | 2004 | β |
| Genetic manipulations of GABAA receptor in mice make inhibition exciting. | Vicini S et al. | β | 2004 | β |
| Imidazo[2,1-b]thiazepines: synthesis, structure and evaluation of benzodiazepine receptor binding. | KieΔ-Kononowicz K et al. | β | 2004 | β |
| Influence of GABAA receptor gamma2 splice variants on receptor kinetics and isoflurane modulation. | Benkwitz C et al. | β | 2004 | β |
| Layer-specific potentiation of evoked IPSCs in rat hippocampal CA1 pyramidal cells by lanthanum. | Kozhemiakin MB et al. | β | 2004 | β |
| Malfunction of respiratory-related neuronal activity in Na+, K+-ATPase alpha2 subunit-deficient mice is attributable to abnormal Cl- homeostasis in brainstem neurons. | Ikeda K et al. | β | 2004 | β |
| Maternal behavior regulates benzodiazepine/GABAA receptor subunit expression in brain regions associated with fear in BALB/c and C57BL/6 mice. | Caldji C et al. | β | 2004 | β |
| Modulation of GABA(A) receptor gene expression by allopregnanolone and ethanol. | Follesa P et al. | β | 2004 | β |
| Modulation of human GABAA and glycine receptor currents by menthol and related monoterpenoids. | Hall AC et al. | β | 2004 | β |
| Multiple structural features of steroids mediate subtype-selective effects on human alpha4beta3delta GABAA receptors. | Pillai GV et al. | β | 2004 | β |
| On the benzodiazepine binding pocket in GABAA receptors. | Berezhnoy D et al. | β | 2004 | β |
| Penicillin blocks human alpha 1 beta 1 and alpha 1 beta 1 gamma 2S GABAA channels that open spontaneously. | Lindquist CE et al. | β | 2004 | β |
| Pharmacological plasticity of GABA(A) receptors at dentate gyrus synapses in a rat model of temporal lobe epilepsy. | Leroy C et al. | β | 2004 | β |
| Positioning of the alpha-subunit isoforms confers a functional signature to gamma-aminobutyric acid type A receptors. | Minier F et al. | β | 2004 | β |
| SB242084, flumazenil, and CRA1000 block ethanol withdrawal-induced anxiety in rats. | Knapp DJ et al. | β | 2004 | β |
| Selective alterations in prefrontal cortical GABA neurotransmission in schizophrenia: a novel target for the treatment of working memory dysfunction. | Lewis DA et al. | β | 2004 | β |
| Studies on the mechanisms of action of picrotoxin, quercetin and pregnanolone at the GABA rho 1 receptor. | Goutman JD et al. | β | 2004 | β |
| Sub-chronic administration of zolpidem affects modifications to rat sleep architecture. | Renger JJ et al. | β | 2004 | β |
| Subregional analysis of GABA(A) receptor subunit mRNAs in the hippocampus of older persons with and without cognitive impairment. | Rissman RA et al. | β | 2004 | β |
| Subunit-specific coupling between gamma-aminobutyric acid type A and P2X2 receptor channels. | BouΓ©-Grabot E et al. | β | 2004 | β |
| The brefeldin A-inhibited GDP/GTP exchange factor 2, a protein involved in vesicular trafficking, interacts with the beta subunits of the GABA receptors. | Charych EI et al. | β | 2004 | β |
| The cerebellar GABAA alpha6 subunit is differentially modulated by chronic ethanol exposure in normal (R100R) and mutated (Q100Q) sNP rats. | Sanna A et al. | β | 2004 | β |
| The interaction of anaesthetic steroids with recombinant glycine and GABAA receptors. | Weir CJ et al. | β | 2004 | β |
| Transcriptional regulation of the mouse gene encoding the alpha-4 subunit of the GABAA receptor. | Ma L et al. | β | 2004 | β |
| Update on PET radiopharmaceuticals: life beyond fluorodeoxyglucose. | Shiue CY et al. | β | 2004 | β |
| Variations in GABRA2, encoding the alpha 2 subunit of the GABA(A) receptor, are associated with alcohol dependence and with brain oscillations. | Edenberg HJ et al. | β | 2004 | β |
| Actions and interactions of extracellular potassium and kainate on expression of 13 gamma-aminobutyric acid type A receptor subunits in cultured mouse cerebellar granule neurons. | Engblom AC et al. | β | 2003 | β |
| Association of GABA(A) receptors and alcohol dependence and the effects of genetic imprinting. | Song J et al. | β | 2003 | β |
| Biochemical analysis of GABA(A) receptor subunits alpha 1, alpha 5, beta 1, beta 2 in the hippocampus of patients with Alzheimer's disease neuropathology. | Rissman RA et al. | β | 2003 | β |
| Changes in GABA(A) receptor gene expression associated with selective alterations in receptor function and pharmacology after ethanol withdrawal. | Sanna E et al. | β | 2003 | β |
| Characterization of wild-type (R100R) and mutated (Q100Q) GABAA alpha 6 subunit in Sardinian alcohol non-preferring rats (sNP). | Sanna A et al. | β | 2003 | β |
| Compartmentation of alpha 1 and alpha 2 GABA(A) receptor subunits within rat extended amygdala: implications for benzodiazepine action. | Kaufmann WA et al. | β | 2003 | β |
| Deletion of the alpha1 or beta2 subunit of GABAA receptors reduces actions of alcohol and other drugs. | Blednov YA et al. | β | 2003 | β |
| Dentate granule cell GABA(A) receptors in epileptic hippocampus: enhanced synaptic efficacy and altered pharmacology. | Cohen AS et al. | β | 2003 | β |
| Diazepam-induced changes on sleep and the EEG spectrum in mice: role of the alpha3-GABA(A) receptor subtype. | Kopp C et al. | β | 2003 | β |
| Distribution of glutamate receptor subunits in experimentally induced cortical malformations. | Hagemann G et al. | β | 2003 | β |
| Dose-dependent EEG effects of zolpidem provide evidence for GABA(A) receptor subtype selectivity in vivo. | Visser SA et al. | β | 2003 | β |
| Drug-induced modification of the system properties associated with spontaneous human electroencephalographic activity. | Liley DT et al. | β | 2003 | β |
| Effects of gamma2S subunit incorporation on GABAA receptor macroscopic kinetics. | Boileau AJ et al. | β | 2003 | β |
| Effects of pentobarbital on GABA-activated currents in acutely-isolated rat dentate gyrus granule neurons. | Lim MS et al. | β | 2003 | β |
| Effects of propofol on GABAA channel conductance in rat-cultured hippocampal neurons. | Eghbali M et al. | β | 2003 | β |
| Evidence for inhibitory effect of the agonist gaboxadol at human alpha 1 beta 2 gamma 2S GABAA receptors. | Smith M et al. | β | 2003 | β |
| Extrasynaptic GABA(A) channels activated by THIP are modulated by diazepam in CA1 pyramidal neurons in the rat brain hippocampal slice. | Lindquist CE et al. | β | 2003 | β |
| Flavonoid modulation of ionic currents mediated by GABA(A) and GABA(C) receptors. | Goutman JD et al. | β | 2003 | β |
| Formation and plasticity of GABAergic synapses: physiological mechanisms and pathophysiological implications. | Fritschy JM et al. | β | 2003 | β |
| GABA(A) alpha1 and alpha2 receptor subunit expression in rostral ventrolateral medulla in nonpregnant and pregnant rats. | Foley CM et al. | β | 2003 | β |
| GABA-A receptor subtypes in the brain: a paradigm for CNS drug discovery? | Whiting PJ | β | 2003 | β |
| Gamma-hydroxybutyric acid and diazepam antagonize a rapid increase in GABA(A) receptors alpha(4) subunit mRNA abundance induced by ethanol withdrawal in cerebellar granule cells. | Follesa P et al. | β | 2003 | β |
| Genetic animal models of anxiety. | Finn DA et al. | β | 2003 | β |
| Heat loss, sleepiness, and impaired performance after diazepam administration in humans. | Echizenya M et al. | β | 2003 | β |
| High affinity central benzodiazepine receptor ligands. Part 3: insights into the pharmacophore and pattern recognition study of intrinsic activities of pyrazolo[4,3-c]quinolin-3-ones. | Carotti A et al. | β | 2003 | β |
| Identified sources and targets of slow inhibition in the neocortex. | TamΓ‘s G et al. | β | 2003 | β |
| Individual properties of the two functional agonist sites in GABA(A) receptors. | Baumann SW et al. | β | 2003 | β |
| Molecular and physiological evidence for functional gamma-aminobutyric acid (GABA)-C receptors in growth hormone-secreting cells. | Gamel-Didelon K et al. | β | 2003 | β |
| Molecular characterization of new polymorphisms at the beta2, alpha1, gamma2 GABA(A) receptor subunit genes associated to a rat nonpreferring ethanol phenotype. | Congeddu E et al. | β | 2003 | β |
| Molecular mechanisms of tolerance to and withdrawal of GABA(A) receptor modulators. | Biggio G et al. | β | 2003 | β |
| Neuroadaptive processes in GABAergic and glutamatergic systems in benzodiazepine dependence. | Allison C et al. | β | 2003 | β |
| Neurosteroid modulation of GABAA receptors. | Lambert JJ et al. | β | 2003 | β |
| Neurosteroids, GABAA receptors, and escalated aggressive behavior. | Miczek KA et al. | β | 2003 | β |
| On high- and low-affinity agonist sites in GABAA receptors. | Baur R et al. | β | 2003 | β |
| Phosphorylation influences neurosteroid modulation of synaptic GABAA receptors in rat CA1 and dentate gyrus neurones. | Harney SC et al. | β | 2003 | β |
| Positron emission tomography radiochemistry. | Mason NS et al. | β | 2003 | β |
| Progesterone withdrawal reduces paired-pulse inhibition in rat hippocampus: dependence on GABA(A) receptor alpha4 subunit upregulation. | Hsu FC et al. | β | 2003 | β |
| Prolonged exposure to gamma-aminobutyric acid up-regulates stably expressed recombinant alpha 1 beta 2 gamma 2s GABAA receptors. | PericiΔ D et al. | β | 2003 | β |
| Radiotracers for positron emission tomography imaging. | Fowler JS et al. | β | 2003 | β |
| Recombinant alpha 1 beta 2 gamma 2 GABA(A) receptors expressed in HEK293 and in QT6 cells show different kinetics. | Mercik K et al. | β | 2003 | β |
| Reducing GABA receptors. | Burt DR | β | 2003 | β |
| Repeated neonatal handling with maternal separation permanently alters hippocampal GABAA receptors and behavioral stress responses. | Hsu FC et al. | β | 2003 | β |
| Rotarod studies in the rat of the GABAA receptor agonist gaboxadol: lack of ethanol potentiation and benzodiazepine cross-tolerance. | Voss J et al. | β | 2003 | β |
| SL651498, a GABAA receptor agonist with subtype-selective efficacy, as a potential treatment for generalized anxiety disorder and muscle spasms. | Griebel G et al. | β | 2003 | β |
| The GABA(A) receptor complex in the chicken brain: immunocytochemical distribution of alpha 1- and gamma 2-subunits and autoradiographic distribution of BZ1 and BZ2 binding sites. | Aller MI et al. | β | 2003 | β |
| The neurobiology and control of anxious states. | Millan MJ | β | 2003 | β |
| The reinforcing properties of alcohol are mediated by GABA(A1) receptors in the ventral pallidum. | June HL et al. | β | 2003 | β |
| The role of GABAA receptors in mediating the effects of alcohol in the central nervous system. | Davies M | β | 2003 | β |
| Thymol, a constituent of thyme essential oil, is a positive allosteric modulator of human GABA(A) receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster. | Priestley CM et al. | β | 2003 | β |
| Variations in maternal care alter GABA(A) receptor subunit expression in brain regions associated with fear. | Caldji C et al. | β | 2003 | β |
| Visualization of alpha5 subunit of GABAA/benzodiazepine receptor by 11C Ro15-4513 using positron emission tomography. | Maeda J et al. | β | 2003 | β |
| 4D-QSAR analysis of a set of propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. | Krasowski MD et al. | β | 2002 | β |
| Acrylamide disturbs the subcellular distribution of GABAA receptor in brain neurons. | Ho WH et al. | β | 2002 | β |
| Affinities of gidazepam and its analogs for mitochondrial benzodiazepine receptors. | Korkhov VM et al. | β | 2002 | β |
| Altered kinetics and benzodiazepine sensitivity of a GABAA receptor subunit mutation [gamma 2(R43Q)] found in human epilepsy. | Bowser DN et al. | β | 2002 | β |
| Altered receptor subtypes in the forebrain of GABA(A) receptor delta subunit-deficient mice: recruitment of gamma 2 subunits. | Korpi ER et al. | β | 2002 | β |
| Benzodiazepine binding studies on living cells: application of small ligands for fluorescence correlation spectroscopy. | Hegener O et al. | β | 2002 | β |
| Bergmann glia GABA(A) receptors concentrate on the glial processes that wrap inhibitory synapses. | Riquelme R et al. | β | 2002 | β |
| Cell type- and input-specific differences in the number and subtypes of synaptic GABA(A) receptors in the hippocampus. | Klausberger T et al. | β | 2002 | β |
| Changes in GABA(A) receptor gene expression induced by withdrawal of, but not by long-term exposure to, zaleplon or zolpidem. | Follesa P et al. | β | 2002 | β |
| Comparison of the effects of zaleplon, zolpidem, and triazolam at various GABA(A) receptor subtypes. | Sanna E et al. | β | 2002 | β |
| Coupled and uncoupled gating and desensitization effects by pore domain mutations in GABA(A) receptors. | Scheller M et al. | β | 2002 | β |
| Differential sensitivity of two insect GABA-gated chloride channels to dieldrin, fipronil and picrotoxinin. | Le Corronc H et al. | β | 2002 | β |
| Different residues in the GABA(A) receptor alpha 1T60-alpha 1K70 region mediate GABA and SR-95531 actions. | Holden JH et al. | β | 2002 | β |
| Drug interactions at GABA(A) receptors. | Korpi ER et al. | β | 2002 | β |
| Early cerebral activities of the environmental estrogen bisphenol A appear to act via the somatostatin receptor subtype sst(2). | Facciolo RM et al. | β | 2002 | β |
| Ectopic expression of the GABA(A) receptor alpha6 subunit in hippocampal pyramidal neurons produces extrasynaptic receptors and an increased tonic inhibition. | Wisden W et al. | β | 2002 | β |
| Effect of flumazenil on GABAA receptors in isolated rat hippocampal neurons. | Weiss M et al. | β | 2002 | β |
| Effects of early postnatal ethanol intubation on GABAergic synaptic proteins. | Hsiao SH et al. | β | 2002 | β |
| Enhanced learning and memory and altered GABAergic synaptic transmission in mice lacking the alpha 5 subunit of the GABAA receptor. | Collinson N et al. | β | 2002 | β |
| Enhanced neurosteroid potentiation of ternary GABA(A) receptors containing the delta subunit. | Wohlfarth KM et al. | β | 2002 | β |
| Forced subunit assembly in alpha1beta2gamma2 GABAA receptors. Insight into the absolute arrangement. | Baumann SW et al. | β | 2002 | β |
| Functional consequences of the loss of high affinity agonist binding to gamma-aminobutyric acid type A receptors. Implications for receptor desensitization. | Newell JG et al. | β | 2002 | β |
| GABA and GABA receptors in the central nervous system and other organs. | Watanabe M et al. | β | 2002 | β |
| GABA(A) receptor beta 2 Tyr97 and Leu99 line the GABA-binding site. Insights into mechanisms of agonist and antagonist actions. | Boileau AJ et al. | β | 2002 | β |
| GABA(A) receptor heterogeneity in histaminergic neurons. | Sergeeva OA et al. | β | 2002 | β |
| GABAergic innervation organizes synaptic and extrasynaptic GABAA receptor clustering in cultured hippocampal neurons. | Christie SB et al. | β | 2002 | β |
| GABA mechanisms and sleep. | Gottesmann C | β | 2002 | β |
| gamma-Aminobutyric acidA rho receptor subunits in the developing rat hippocampus. | Didelon F et al. | β | 2002 | β |
| Gamma-aminobutyric acid transporter (BGT-1) expressed in human astrocytoma U373 MG cells: pharmacological and molecular characterization and phorbol ester-induced inhibition. | Ruiz-TachiquΓn ME et al. | β | 2002 | β |
| Homologous sites of GABA(A) receptor alpha(1), beta(3) and gamma(2) subunits are important for assembly. | Sarto I et al. | β | 2002 | β |
| Localisation of GABA(A) receptor epsilon-subunit in cholinergic and aminergic neurones and evidence for co-distribution with the theta-subunit in rat brain. | Moragues N et al. | β | 2002 | β |
| Mechanism-based pharmacodynamic modeling of the interaction of midazolam, bretazenil, and zolpidem with ethanol. | Tuk B et al. | β | 2002 | β |
| Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors. | Wingrove PB et al. | β | 2002 | β |
| Mechanisms of pyrethroid neurotoxicity: implications for cumulative risk assessment. | Soderlund DM et al. | β | 2002 | β |
| Molecular actions of (S)-desmethylzopiclone (SEP-174559), an anxiolytic metabolite of zopiclone. | Fleck MW | β | 2002 | β |
| Molecular determinants for the action of general anesthetics at recombinant alpha(2)beta(3)gamma(2)gamma-aminobutyric acid(A) receptors. | Siegwart R et al. | β | 2002 | β |
| Neonatal toluene exposure selectively alters sensitivity to different chemoconvulsant drugs in juvenile rats. | Chen HH et al. | β | 2002 | β |
| Neuroactive steroid mechanisms and GABA type A receptor subunit assembly in hypothalamic and extrahypothalamic regions. | Canonaco M et al. | β | 2002 | β |
| Neuronal activity and its influence on developmentally regulated GABA(A) receptor expression in cultured mouse cerebellar granule cells. | Ives JH et al. | β | 2002 | β |
| Pathophysiological aspects of diversity in neuronal inhibition: a new benzodiazepine pharmacology. | MΓΆhler H | β | 2002 | β |
| Pharmacological characterization of a novel cell line expressing human alpha(4)beta(3)delta GABA(A) receptors. | Brown N et al. | β | 2002 | β |
| Pharmacological characterization of a novel cell line expressing human alpha(4)beta(3)delta GABA(A) receptors: commentary on Brown et al. | Lambert JJ et al. | β | 2002 | β |
| Pharmacological heterogeneity of gamma-aminobutyric acid receptors during development suggests distinct classes of rat cerebellar granule cells in situ. | Hevers W et al. | β | 2002 | β |
| Propofol enhances GABA(A) receptor-mediated presynaptic inhibition in human spinal cord. | Shimizu M et al. | β | 2002 | β |
| Quantitative reverse transcription-polymerase chain reaction of GABA(A) alpha1, beta1 and gamma2S subunits in epileptic rats following photothrombotic infarction of neocortex. | Liu J et al. | β | 2002 | β |
| Relative picrotoxin insensitivity distinguishes ionotropic GABA receptor-mediated IPSCs in hippocampal interneurons. | Semyanov A et al. | β | 2002 | β |
| Release-independent short-term facilitation at GABAergic synapses in the olfactory bulb. | Nusser Z | β | 2002 | β |
| Role of the histidine residue at position 105 in the human alpha 5 containing GABA(A) receptor on the affinity and efficacy of benzodiazepine site ligands. | Kelly MD et al. | β | 2002 | β |
| Synaptic and extrasynaptic GABAA receptor and gephyrin clusters. | Christie SB et al. | β | 2002 | β |
| The 5'-flanking region of the rat GABA(A) receptor alpha2-subunit gene (Gabra2). | Fuchs K et al. | β | 2002 | β |
| The beta-lactam antibiotics, penicillin-G and cefoselis have different mechanisms and sites of action at GABA(A) receptors. | Sugimoto M et al. | β | 2002 | β |
| Tracazolate reveals a novel type of allosteric interaction with recombinant gamma-aminobutyric acid(A) receptors. | Thompson SA et al. | β | 2002 | β |
| Truncation of the GABA(A)-receptor gamma2 subunit in a family with generalized epilepsy with febrile seizures plus. | Harkin LA et al. | β | 2002 | β |
| Unique assignment of inter-subunit association in GABA(A) alpha 1 beta 3 gamma 2 receptors determined by molecular modeling. | Trudell J | β | 2002 | β |
| Volatile anesthetic actions on the GABAA receptors: contrasting effects of alpha 1(S270) and beta 2(N265) point mutations. | Nishikawa K et al. | β | 2002 | β |
| [3H]Flunitrazepam binding to recombinant alpha1beta2gamma2S GABAA receptors stably expressed in HEK 293 cells. | PericiΔ D et al. | β | 2001 | β |
| Activation of GABA(A) receptors in subthalamic neurons in vitro: properties of native receptors and inhibition mechanisms. | Baufreton J et al. | β | 2001 | β |
| Altered atypical coupling of gamma-aminobutyrate type A receptor agonist and convulsant binding sites in subunit-deficient mouse lines. | Sinkkonen ST et al. | β | 2001 | β |
| Alternate use of distinct intersubunit contacts controls GABAA receptor assembly and stoichiometry. | Klausberger T et al. | β | 2001 | β |
| Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABA(A) receptors. | Ebert B et al. | β | 2001 | β |
| Changes in the gene expression of GABA(A) receptor alpha1 and alpha2 subunits and metabotropic glutamate receptor 5 in the basal ganglia of the rats with unilateral 6-hydroxydopamine lesion and embryonic mesencephalic grafts. | Yu TS et al. | β | 2001 | β |
| Characterization of gamma-aminobutyrate type A receptors with atypical coupling between agonist and convulsant binding sites in discrete brain regions. | Sinkkonen ST et al. | β | 2001 | β |
| Chronic prenatal ethanol exposure increases GABA(A) receptor subunit protein expression in the adult guinea pig cerebral cortex. | Bailey CD et al. | β | 2001 | β |
| Common effects of chronically administered antipanic drugs on brainstem GABA(A) receptor subunit gene expression. | Tanay VM et al. | β | 2001 | β |
| Detection and binding properties of GABA(A) receptor assembly intermediates. | Klausberger T et al. | β | 2001 | β |
| Differential cross talk of ROD compounds with the benzodiazepine binding site. | Sigel E et al. | β | 2001 | β |
| Differentiation of GABA(A) receptors in subcortical heterotopias: subunit distribution of displaced cortex reflects original commitment. | Hagemann G et al. | β | 2001 | β |
| Do antiepileptics phenytoin, carbamazepine, and loreclezole show GABA(A) receptor subtype selectivity in rat brain sections? | Holopainen IE et al. | β | 2001 | β |
| Effect of embryonic knock-down of GABAA receptors on the levels of monoamines and their metabolites in the CNS of the mouse. | Ugarte SD et al. | β | 2001 | β |
| Effects of gamma-HCH and delta-HCH on human recombinant GABA(A) receptors: dependence on GABA(A) receptor subunit combination. | Maskell PD et al. | β | 2001 | β |
| Epilepsy-associated plasticity in gamma-aminobutyric acid receptor expression, function, and inhibitory synaptic properties. | Coulter DA | β | 2001 | β |
| Fipronil-based photoaffinity probe for Drosophila and human beta 3 GABA receptors. | Sirisoma NS et al. | β | 2001 | β |
| Functional pharmacology of GABA(A) receptors containing the chicken brain gamma 4 subunit. | Forster IC et al. | β | 2001 | β |
| GABA(A)-receptor delta subunit knockout mice have multiple defects in behavioral responses to ethanol. | Mihalek RM et al. | β | 2001 | β |
| GABAA-receptor plasticity during long-term exposure to and withdrawal from progesterone. | Biggio G et al. | β | 2001 | β |
| GABA(A) receptor subtypes: dissecting their pharmacological functions. | Rudolph U et al. | β | 2001 | β |
| GABA(B) receptor activation enhances mGluR-mediated responses at cerebellar excitatory synapses. | Hirono M et al. | β | 2001 | β |
| gamma-Aminobutyric acid(A) receptor subunit expression predicts functional changes in hippocampal dentate granule cells during postnatal development. | Brooks-Kayal AR et al. | β | 2001 | β |
| Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor. | Casula MA et al. | β | 2001 | β |
| Increase in expression of the GABA(A) receptor alpha(4) subunit gene induced by withdrawal of, but not by long-term treatment with, benzodiazepine full or partial agonists. | Follesa P et al. | β | 2001 | β |
| Inhibitory effect of theophylline on recombinant GABA(A) receptor. | Sugimoto T et al. | β | 2001 | β |
| Input-dependent synaptic targeting of alpha(2)-subunit-containing GABA(A) receptors in synapses of hippocampal pyramidal cells of the rat. | NyΓri G et al. | β | 2001 | β |
| Loss of the major GABA(A) receptor subtype in the brain is not lethal in mice. | Sur C et al. | β | 2001 | β |
| Magnesium potentiation of the function of native and recombinant GABA(A) receptors. | MΓΆykkynen T et al. | β | 2001 | β |
| Modulation of native and recombinant GABA(A) receptors by endogenous and synthetic neuroactive steroids. | Lambert JJ et al. | β | 2001 | β |
| Molecular and cellular properties of GnRH neurons revealed through transgenics in the mouse. | Herbison AE et al. | β | 2001 | β |
| Molecular modeling and QSAR analysis of the interaction of flavone derivatives with the benzodiazepine binding site of the GABA(A) receptor complex. | Marder M et al. | β | 2001 | β |
| Morphine withdrawal increases expression of GABA(A) receptor epsilon subunit mRNA in locus coeruleus neurons. | HeikkilΓ€ AT et al. | β | 2001 | β |
| Mutagenesis of the GABA(A) receptor alpha1 subunit reveals a domain that affects sensitivity to GABA and benzodiazepine-site ligands. | Davies M et al. | β | 2001 | β |
| Neurosteroid modulation of recombinant and synaptic GABAA receptors. | Lambert JJ et al. | β | 2001 | β |
| New insights into the role of the GABA(A)-benzodiazepine receptor in psychiatric disorder. | Nutt DJ et al. | β | 2001 | β |
| Nitric oxide directly activates GABA(A) receptor function through a cGMP/protein kinase-independent pathway in frog pituitary melanotrophs. | Castel H et al. | β | 2001 | β |
| Non-competitive GABA antagonists: probing the mechanisms of their selectivity for insect versus mammalian receptors. | Ozoe Y et al. | β | 2001 | β |
| Pathway-specific targeting of GABA(A) receptor subtypes to somatic and dendritic synapses in the central amygdala. | Delaney AJ et al. | β | 2001 | β |
| Physiological roles for the neurosteroid allopregnanolone in the modulation of brain function during pregnancy and parturition. | Herbison AE | β | 2001 | β |
| Postnatal maturation of human GABAA receptors measured with positron emission tomography. | Chugani DC et al. | β | 2001 | β |
| Regulation of the subcellular distribution and gene expression of GABA(A) receptor by microtubules and microfilaments in cultured brain neurons. | Ho WH et al. | β | 2001 | β |
| Role of allopregnanolone in regulation of GABA(A) receptor plasticity during long-term exposure to and withdrawal from progesterone. | Follesa P et al. | β | 2001 | β |
| Role of human GABA(A) receptor beta3 subunit in insecticide toxicity. | Ratra GS et al. | β | 2001 | β |
| Structure and function of GABA(C) receptors: a comparison of native versus recombinant receptors. | Zhang D et al. | β | 2001 | β |
| The GABA(A) Receptor: Subunit-Dependent Functions and Absence Seizures. | Wong CG et al. | β | 2001 | β |
| The KCl cotransporter, KCC2, is highly expressed in the vicinity of excitatory synapses in the rat hippocampus. | GulyΓ‘s AI et al. | β | 2001 | β |
| The R100Q mutation of the GABA(A) alpha(6) receptor subunit may contribute to voluntary aversion to ethanol in the sNP rat line. | Saba L et al. | β | 2001 | β |
| Two novel residues in M2 of the gamma-aminobutyric acid type A receptor affecting gating by GABA and picrotoxin affinity. | Buhr A et al. | β | 2001 | β |
| Abuse, dependence, and epileptic seizures after zolpidem withdrawal: review and case report. | Aragona M | β | 2000 | β |
| Allosteric modulators affect the efficacy of partial agonists for recombinant GABA(A) receptors. | Maksay G et al. | β | 2000 | β |
| (+)- and (-)-cis-2-aminomethylcyclopropanecarboxylic acids show opposite pharmacology at recombinant rho(1) and rho(2) GABA(C) receptors. | Duke RK et al. | β | 2000 | β |
| Anion transport in heart. | Hume JR et al. | β | 2000 | β |
| A novel positive allosteric modulator of the GABA(A) receptor: the action of (+)-ROD188. | Thomet U et al. | β | 2000 | β |
| Applications of transgenic and knockout mice in alcohol research. | Bowers BJ | β | 2000 | β |
| A single glycine residue at the entrance to the first membrane-spanning domain of the gamma-aminobutyric acid type A receptor beta(2) subunit affects allosteric sensitivity to GABA and anesthetics. | Carlson BX et al. | β | 2000 | β |
| Behavioural effects of a benzodiazepine receptor partial agonist, Ro 19-8022, in the social conflict test in mice. | Podhorna J et al. | β | 2000 | β |
| Benzodiazepines act on GABAA receptors via two distinct and separable mechanisms. | Walters RJ et al. | β | 2000 | β |
| Benzodiazepine-sensitive GABA(A) receptors limit the activity of the NMDA/NO/cyclic GMP pathway: a microdialysis study in the cerebellum of freely moving rats. | Fedele E et al. | β | 2000 | β |
| Bicuculline, pentobarbital and diazepam modulate spontaneous GABA(A) channels in rat hippocampal neurons. | Birnir B et al. | β | 2000 | β |
| Characterization of the interaction of zopiclone with gamma-aminobutyric acid type A receptors. | Davies M et al. | β | 2000 | β |
| Coexpression of rat P2X2 and P2X6 subunits in Xenopus oocytes. | King BF et al. | β | 2000 | β |
| Coupling between agonist and chloride ionophore sites of the GABA(A) receptor: agonist/antagonist efficacy of 4-PIOL. | Rabe H et al. | β | 2000 | β |
| Differential downregulation of GABAA receptor subunits in widespread brain regions in the freeze-lesion model of focal cortical malformations. | Redecker C et al. | β | 2000 | β |
| Differential modulatory actions of the volatile convulsant flurothyl and its anesthetic isomer at inhibitory ligand-gated ion channels. | Krasowski MD | β | 2000 | β |
| Direct protein-protein coupling enables cross-talk between dopamine D5 and gamma-aminobutyric acid A receptors. | Liu F et al. | β | 2000 | β |
| Early expression of GABA(A) receptor delta subunit in the neonatal rat hippocampus. | Didelon F et al. | β | 2000 | β |
| Electrophysiological evidence for the coexistence of alpha1 and alpha6 subunits in a single functional GABA(A) receptor. | Sigel E et al. | β | 2000 | β |
| Epilepsy genes: the link between molecular dysfunction and pathophysiology. | Stafstrom CE et al. | β | 2000 | β |
| GABA(A)-mediated toxicity of hippocampal neurons in vitro. | Lukasiuk K et al. | β | 2000 | β |
| GABA(A) receptor assembly. Identification and structure of gamma(2) sequences forming the intersubunit contacts with alpha(1) and beta(3) subunits. | Klausberger T et al. | β | 2000 | β |
| GABA(A) receptor epsilon and theta subunits display unusual structural variation between species and are enriched in the rat locus ceruleus. | Sinkkonen ST et al. | β | 2000 | β |
| GABAC receptors are localized with microtubule-associated protein 1B in mammalian cone photoreceptors. | Pattnaik B et al. | β | 2000 | β |
| GABA potentiation: a logical pharmacological approach for the treatment of acute ischaemic stroke. | Green AR et al. | β | 2000 | β |
| Genetic inactivation of the Serotonin(1A) receptor in mice results in downregulation of major GABA(A) receptor alpha subunits, reduction of GABA(A) receptor binding, and benzodiazepine-resistant anxiety. | Sibille E et al. | β | 2000 | β |
| Harmaline-induced changes in gamma aminobutyric acid(A) receptor subunit mRNA expression in murine olivocerebellar nuclei. | Frostholm A et al. | β | 2000 | β |
| Late postnatal reorganization of GABA(A) receptor signalling in native GnRH neurons. | Sim JA et al. | β | 2000 | β |
| Long-range interactions in neuronal gene expression: evidence from gene targeting in the GABA(A) receptor beta2-alpha6-alpha1-gamma2 subunit gene cluster. | Uusi-Oukari M et al. | β | 2000 | β |
| Modulation of GABA(A) receptor subunit mRNA levels in olivocerebellar neurons of purkinje cell degeneration and weaver mutant mice. | Rotter A et al. | β | 2000 | β |
| Neurochemical and metabolic aspects of antidepressants: an overview. | Baker GB et al. | β | 2000 | β |
| Neurochemical and molecular pharmacological aspects of the GABA(B) receptor. | Kuriyama K et al. | β | 2000 | β |
| New benzodiazepines alter acetylcholinesterase and ATPDase activities. | Schetinger MR et al. | β | 2000 | β |
| Non-coordinate regulation of endogenous epithelial sodium channel (ENaC) subunit expression at the apical membrane of A6 cells in response to various transporting conditions. | Weisz OA et al. | β | 2000 | β |
| Pentobarbital modulates gamma-aminobutyric acid-activated single-channel conductance in rat cultured hippocampal neurons. | Eghbali M et al. | β | 2000 | β |
| Pharmacology of AMPA/kainate receptor ligands and their therapeutic potential in neurological and psychiatric disorders. | Lees GJ | β | 2000 | β |
| Pharmacology of GABA(A) receptors of retinal dopaminergic neurons. | Feigenspan A et al. | β | 2000 | β |
| Quantification of GABA(A) receptor subunit mRNAs by non-radioisotopic competitive RT-PCR utilizing plate-based EIA methodology. | Uusi-Oukari M et al. | β | 2000 | β |
| Role of the GABA(A)beta2, GABA(A)alpha6, GABA(A)alpha1 and GABA(A)gamma2 receptor subunit genes cluster in drug responses and the development of alcohol dependence. | Loh EW et al. | β | 2000 | β |
| Role of the GABA(A) receptor gamma2 subunit in the development of gonadotropin-releasing hormone neurons in vivo. | Simonian SX et al. | β | 2000 | β |
| Sedative but not anxiolytic properties of benzodiazepines are mediated by the GABA(A) receptor alpha1 subtype. | McKernan RM et al. | β | 2000 | β |
| Selective alterations in GABAA receptor subtypes in human temporal lobe epilepsy. | Loup F et al. | β | 2000 | β |
| Sh and eag K(+) channel subunit interaction in frog oocytes depends on level and time of expression. | Chen ML et al. | β | 2000 | β |
| Single-channel properties of neuronal GABAA receptors from mice lacking the 2 subunit. | Lorez M et al. | β | 2000 | β |
| The actions of ether, alcohol and alkane general anaesthetics on GABAA and glycine receptors and the effects of TM2 and TM3 mutations. | Krasowski MD et al. | β | 2000 | β |
| The alpha and gamma subunit-dependent effects of local anesthetics on recombinant GABA(A) receptors. | Sugimoto M et al. | β | 2000 | β |
| The triakontatetraneuropeptide (TTN) stimulates thymidine incorporation in rat astrocytes through peripheral-type benzodiazepine receptors. | Gandolfo P et al. | β | 2000 | β |
| Tryptophan scanning mutagenesis in TM2 of the GABA(A) receptor alpha subunit: effects on channel gating and regulation by ethanol. | Ueno S et al. | β | 2000 | β |
| Unraveling the function of GABA(A) receptor subtypes. | Sieghart W | β | 2000 | β |
| Use of bicuculline, a GABA antagonist, as a template for the development of a new class of ligands showing positive allosteric modulation of the GABA(A) receptor. | Razet R et al. | β | 2000 | β |
| Altered GABA(A)-benzodiazepine receptor number and pharmacology in the adult guinea pig cerebral cortex after chronic prenatal ethanol exposure. | Bailey CD et al. | β | 1999 | β |
| An in situ hybridization study of the distribution of the GABA(B2) protein mRNA in the rat CNS. | Durkin MM et al. | β | 1999 | β |
| An update on GABAA receptors. | Mehta AK et al. | β | 1999 | β |
| A significant part of native gamma-aminobutyric AcidA receptors containing alpha4 subunits do not contain gamma or delta subunits. | Bencsits E et al. | β | 1999 | β |
| A single amino acid confers barbiturate sensitivity upon the GABA rho 1 receptor. | Belelli D et al. | β | 1999 | β |
| A single amino acid in the second transmembrane domain of GABA rho subunits is a determinant of the response kinetics of GABAC receptors. | Qian H et al. | β | 1999 | β |
| Attenuated sensitivity to neuroactive steroids in gamma-aminobutyrate type A receptor delta subunit knockout mice. | Mihalek RM et al. | β | 1999 | β |
| Benzodiazepine actions mediated by specific gamma-aminobutyric acid(A) receptor subtypes. | Rudolph U et al. | β | 1999 | β |
| Composition of the GABA(A) receptors of retinal dopaminergic neurons. | Gustincich S et al. | β | 1999 | β |
| Differential effects of zinc on native GABA(A) receptor function in rat hippocampus and cerebellum. | Schmid G et al. | β | 1999 | β |
| Differential regulation of synaptic GABAA receptors by cAMP-dependent protein kinase in mouse cerebellar and olfactory bulb neurones. | Nusser Z et al. | β | 1999 | β |
| Effect of pirenzepine, a muscarinic M1 receptor antagonist, on amygdala kindling in rat. | EΕkazan E et al. | β | 1999 | β |
| Effect of surgical stress on benzodiazepine receptors as a consequence of placebo pellet implantation in rat: an autoradiographic study. | Revilla V et al. | β | 1999 | β |
| Enhanced benzodiazepine and ethanol actions on cerebellar GABA(A) receptors mediating glutamate release in an alcohol-sensitive rat line. | Schmid G et al. | β | 1999 | β |
| Evaluation of [methyl-3H]L655,708 and [ethyl-3H]RY80 as putative PET ligands for central GABA(A) receptors containing alpha5 subunit. | Opacka-Juffry J et al. | β | 1999 | β |
| GABA receptors inhibited by benzodiazepines mediate fast inhibitory transmission in the central amygdala. | Delaney AJ et al. | β | 1999 | β |
| General anaesthetic action at transmitter-gated inhibitory amino acid receptors. | Belelli D et al. | β | 1999 | β |
| General anaesthetic actions on ligand-gated ion channels. | Krasowski MD et al. | β | 1999 | β |
| Hetero-oligomeric assembly of P2X receptor subunits. Specificities exist with regard to possible partners. | Torres GE et al. | β | 1999 | β |
| Human neuronal gamma-aminobutyric acid(A) receptors: coordinated subunit mRNA expression and functional correlates in individual dentate granule cells. | Brooks-Kayal AR et al. | β | 1999 | β |
| Identification of a domain involved in ATP-gated ionotropic receptor subunit assembly. | Torres GE et al. | β | 1999 | β |
| Identification of subunits mediating clustering of GABA(A) receptors by rapsyn. | Ebert V et al. | β | 1999 | β |
| Identification of transduction elements for benzodiazepine modulation of the GABA(A) receptor: three residues are required for allosteric coupling. | Boileau AJ et al. | β | 1999 | β |
| Indoleamine-accumulating amacrine cells are presynaptic to rod bipolar cells through GABA(C) receptors. | Fletcher EL et al. | β | 1999 | β |
| Mapping quantitative trait loci for seizure response to a GABAA receptor inverse agonist in mice. | Gershenfeld HK et al. | β | 1999 | β |
| Mapping the agonist binding site of the GABAA receptor: evidence for a beta-strand. | Boileau AJ et al. | β | 1999 | β |
| Postnatal ethanol exposure blunts upregulation of GABAA receptor currents in Purkinje neurons. | Hsiao SH et al. | β | 1999 | β |
| Response kinetics and pharmacological properties of heteromeric receptors formed by coassembly of GABA rho- and gamma 2-subunits. | Qian H et al. | β | 1999 | β |
| Role of GABAA and GABAC receptors in the biphasic GABA responses in neurons of the rat major pelvic ganglia. | Akasu T et al. | β | 1999 | β |
| Single-channel properties of synaptic and extrasynaptic GABAA receptors suggest differential targeting of receptor subtypes. | Brickley SG et al. | β | 1999 | β |
| Structure and subunit composition of GABA(A) receptors. | Sieghart W et al. | β | 1999 | β |
| The intrinsic specification of gamma-aminobutyric acid type A receptor alpha6 subunit gene expression in cerebellar granule cells. | Bahn S et al. | β | 1999 | β |
| Towards better benzodiazepines. | Wisden W et al. | β | 1999 | β |
| The Pharmacology and Mechanism of Action of Zolpidem. | Sanger DJ et al. | β | 1998 | β |